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JWH-030: Wikis

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JWH-030
Systematic (IUPAC) name
naphthalen-1-yl-(1-pentylpyrrol- 3-yl)methanone
Identifiers
CAS number 162934-73-8
ATC code  ?
PubChem 9971539
Chemical data
Formula C 20H21NO 
Mol. mass 291.386 g/mol
SMILES eMolecules & PubChem
Pharmacokinetic data
Bioavailability  ?
Metabolism  ?
Half life  ?
Excretion  ?
Therapeutic considerations
Pregnancy cat.  ?
Legal status
Routes  ?

JWH-030 is a drug which is a cannabinoid receptor agonist.[1] It has analgesic effects and is used in scientific research.[2] It is a partial agonist at CB1 receptors, with a Ki of 87nM, making it roughly half the potency of THC.[3]

References

  1. ^ Lainton JAH, Huffman JW, Martin BR, Compton DR. Tetrahedron Letters. 1995; 36:1401.
  2. ^ Pertwee RG, Griffin, G, Lainton JAH, Huffman JW. European Journal of Pharmacology. 1995; 284:241.
  3. ^ Griffin, G; Atkinson; Showalter; Martin; Abood (1998). "Evaluation of cannabinoid receptor agonists and antagonists using the guanosine-5'-O-(3-35Sthio)-triphosphate binding assay in rat cerebellar membranes". The Journal of pharmacology and experimental therapeutics 285 (2): 553–60. PMID 9580597.   edit
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